CPI-1205 25mL Class A

CPI-1205 25mL Class ACPI 1205 is an orally available selective inhibitor of the histone lysine methyltransferase EZH2 with IC50 values of 2 nM and 52 nM for EZH2 and EZH1 respectively. It has potential antineoplastic activity.

Dicoumarol is a competitive NADPH quinone oxidoreductase (NQO1) inhibitor

2-Aminobenzenesulfonamide is an inhibitor of carbonic anhydrase IX

Kynurenic acid

Corning The capacity tolerance on this Class A 100mL PYREX® buret is established by ASTM E-287 and is calibrated in accordance with ASTM E-542

an inhibitor of tetrahydrofolate dehydrogenase

SH2) and PTP1B

-induced PAI-1 overexpression via extracellular signal-related kinases (ERK1/2) and phosphatidylinositol 3-kinase (PI3K)/protein kinase B (PKB) signaling pathways

Inhibits ATR with IC50 of 21 nM in 3T3TopBP1-ER cell

PXR and FXR

9 nM and 1

Euphorbiasteroid

Now for the heavy lifting